Synthesis and acaricidal activity of strobilurin-pyrimidine derivatives
查看参考文献16篇
文摘
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Pyriminostrobin, a new acaricide, was discovered in our previous studies. Because introducing fluorine into organic compounds can increase bioactivity, pyriminostrobin was modified as a series of strobilurin-pyrimidine derivatives for biological screening. The compounds were characterized by~1H NMR, MS and elemental analysis. Preliminary bioassays demonstrated that compounds 7e and 7i exhibited significant control against Tetranychus cinnabarinus (Boisd.) at 0.625 mg L~(-10, and their acaricidal potencies were higher than pyriminostrobin in a greenhouse. The relationship between structure and acaricidal activity was also studied. |
来源
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Chinese Chemical Letters
,2014,25(1):137-140 【核心库】
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DOI
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10.1016/j.cclet.2013.10.006
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关键词
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Strobilurin-pyrimidine
;
Acaricidal activity
;
Intermediate derivatization method
;
Pyriminostrobin
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地址
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1.
College of Chemistry and Molecular Engineering, Zhengzhou University,, State Key Laboratory of the Discovery and Development of Novel Pesticide, Zhengzhou, 450001
2.
Shenyang Research Institute of Chemical Industry Co., Ltd., State Key Laboratory of the Discovery and Development of Novel Pesticide, Shenyang, 110021
3.
College of Chemistry and Molecular Engineering, Zhengzhou University,, Zhengzhou, 450001
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语种
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英文 |
文献类型
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研究性论文 |
ISSN
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1001-8417 |
学科
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化学 |
基金
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the Outstanding Young Scholarship from the National Natural Science Foundation of China
;
国家自然科学基金
;
the Outstanding Scholar Foundation of Henan Province
;
supported by the National Key Basic Research Program of China (973 Program)
;
the National Key Technology Support Program during the 12th Five-Year Plan Period
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文献收藏号
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CSCD:5050814
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