Design, synthesis, and fungicidal activity of novel 1,3,4-oxadiazole derivatives
查看参考文献34篇
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文摘
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Employing the intermediate derivatization method (IDM), twenty novel 1,3,4-oxadiazole derivatives containing arylpyrazoloxyl moietywere designed and synthesized. The structures of the title compounds were identified by ~1H NMR, ~(13)C NMR, MS and elemental analyses, compound 4 was further identified by single-crystal X-ray diffraction. Antifungal activities against rice sheath blight (RSB)and sorghum anthracnose (SA)were evaluated by the mycelium linear growth rate method. Compounds 4, 16 and 20 displayed significant activities against RSB (EC_(50) = 0.88 mg/L, 0.91 mg/L and 0.85 mg/L, respectively), higher than the reference tebuconazole; While compound 3 exhibited higher activity against SA (EC_(50) = 1.03 mg/L), equal to commercial pyraclostrobin (EC_(50) = 1.06 mg/L). The study showed that compound 20 is a promising fungicide for further development. |
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来源
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Chinese Chemical Letters
,2018,29(6):915-918 【核心库】
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DOI
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10.1016/j.cclet.2018.01.050
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关键词
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1,3,4-Oxadiazole derivatives
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Intermediate derivatization method
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Rice sheath blight
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Sorghum anthracnose
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Structure-activity relationship
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地址
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1.
Department of Materials Physics and Chemistry,School of Material Science and Engineering,,Northeastern University, Key Laboratory for Anisotropy and Texture of Materials,Ministry of Education, Shenyang, 110819
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Shenyang Sinochem Agrochemicals R&D Co.,Ltd., State Key Laboratory of the Discovery and Development of Novel Pesticide, Shenyang, 110021
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语种
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英文 |
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文献类型
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综述型 |
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ISSN
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1001-8417 |
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学科
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化学工业 |
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基金
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supported partially by the Open Foundation of Key Laboratory for Anisotropy and Texture of Materials, Ministry of Education, Northeastern University, China
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文献收藏号
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CSCD:6275686
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引证文献
2
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1
Yu Fuqiang
Design, Synthesis and Fungicidal Activity against Rhizoctonia solani of New Phenylpyrazoloxyl Propionic Acid Derivatives
有机化学,2019,39(2):397-405
CSCD被引
0
次
2
He Min
Design, synthesis and fungicidal activities of phenazine-1-carboxamida conjugates of 1,3,4-thia(oxa)diazole
农药学学报,2021,23(2):287-295
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0
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