帮助 关于我们

返回检索结果

Synthesis and acaricidal activity of strobilurin-pyrimidine derivatives

查看参考文献16篇

文摘 Pyriminostrobin, a new acaricide, was discovered in our previous studies. Because introducing fluorine into organic compounds can increase bioactivity, pyriminostrobin was modified as a series of strobilurin-pyrimidine derivatives for biological screening. The compounds were characterized by~1H NMR, MS and elemental analysis. Preliminary bioassays demonstrated that compounds 7e and 7i exhibited significant control against Tetranychus cinnabarinus (Boisd.) at 0.625 mg L~(-10, and their acaricidal potencies were higher than pyriminostrobin in a greenhouse. The relationship between structure and acaricidal activity was also studied.
来源 Chinese Chemical Letters ,2014,25(1):137-140 【核心库】
DOI 10.1016/j.cclet.2013.10.006
关键词 Strobilurin-pyrimidine ; Acaricidal activity ; Intermediate derivatization method ; Pyriminostrobin
地址

1. College of Chemistry and Molecular Engineering, Zhengzhou University,, State Key Laboratory of the Discovery and Development of Novel Pesticide, Zhengzhou, 450001  

2. Shenyang Research Institute of Chemical Industry Co., Ltd., State Key Laboratory of the Discovery and Development of Novel Pesticide, Shenyang, 110021  

3. College of Chemistry and Molecular Engineering, Zhengzhou University,, Zhengzhou, 450001

语种 英文
文献类型 研究性论文
ISSN 1001-8417
学科 化学
基金 the Outstanding Young Scholarship from the National Natural Science Foundation of China ;  国家自然科学基金 ;  the Outstanding Scholar Foundation of Henan Province ;  supported by the National Key Basic Research Program of China (973 Program) ;  the National Key Technology Support Program during the 12th Five-Year Plan Period
文献收藏号 CSCD:5050814

参考文献 共 16 共1页

1.  Chai B S. The discovery of SYP-10913 and SYP-11277: novel strobilurin acaricides. Pest Manag. Sci,2011,67:1141-1146 被引 5    
2.  Chai B S. The discovery of acaricide SYP-11277. Agrochemical(in Chinese),2011,5:325-326 被引 1    
3.  Liu C L. New agrochemical candidates from intermediate derivatization method based on bioisosteric replacement. Frontiers of Modern Chem ical Engineering, Metallurgy, and Material Technologies-7th Academic Conference of Chemical, Metallurgy and Material Engineering Department, CAE,2009:86-94 被引 1    
4.  Liu C L. Innovation of pesticide discovery methods and candidate compounds. High-Technol. Ind (Chinese),2008,9:79-81 被引 2    
5.  Liu C L. New approach for agrochemical discovery and application (1)-intermediate derivatization method. Agrochemical (in Chinese),2011,1:20-22 被引 2    
6.  Dolbier W R. Fluorine chemistry at the millennium. J. Fluorine Chem,2005,126:157-163 被引 6    
7.  El-Sharief M A. Synthesis, characterization, and derivatization of some novel types of fluorinated mono-and bis-imidazolidineiminothiones with antitumor, antiviral, antibacterial, and antifungal activities. J. Fluorine Chem,2011,132:596-611 被引 1    
8.  Liu A P. Synthesis and fungicidal activities of novel bis(trifluoromethyl)phenyl-based strobilurins. J. Agric. Food Chem,2008,56:6562-6566 被引 3    
9.  Liu A P. The discovery of HNPC-A3066: a novel strobilurin acaricide. Pest Manag. Sci,2008,65:229-234 被引 1    
10.  Faidallah H M. Synthesis and biological evaluation of new 3,5-di(trifluoromethyl)-1,2,4-triazolesulfonylurea and thiourea derivatives as antidiabetic and antimicrobial agents. J. Fluorine Chem,2011,132:870-877 被引 1    
11.  Li S. Synthesis and fungicidal activity of new fluorinecontainingmandelic acid amide compounds. J. Fluorine Chem,2012,137:108-112 被引 3    
12.  Saeed A. Synthesis and antimicrobial activity of some novel 2-(substituted fluorobenzoylimino)-3-(substituted fluorophenyl)-4-methyl-1,3-thiazolines. J. Fluorine Chem,2010,131:333-339 被引 1    
13.  Li H C. Synthesis and fungicidal activity of novel strobilurin analogues containing substituted N-phenylpyrimidin-2-amines. Chin. Chem. Lett,2009,20:1287-1290 被引 3    
14.  Chai B S. Design, synthesis and acaricidal activity of novel strobilurin derivatives containing pyrimidine moieties. Pest Manag. Sci,2010,66:1208-1214 被引 5    
15.  Harada K. Coumarins as novel17b-hydroxysteroid dehydrogenase type 3 inhibitors for potential treatment of prostate cancer. Bioorg. Med. Chem. Lett,2010,20:272-275 被引 2    
16.  Tomlin C D S. Fluacrypyrim. The Pesticide Manual (14th ed),2006:471-472 被引 1    
引证文献 3

1 陈美航 嘧啶类衍生物的杀虫活性研究新进展 农药,2018,57(12):859-863
被引 1

2 Cao Yangyang Synthesis and Herbicidal Activity of Novel β-Methoxyacrylate Derivatives Containing a Substituted Phenylpyridine Moiety Chemical Research in Chinese Universities,2019,35(6):1008-1011
被引 0 次

显示所有3篇文献

论文科学数据集
PlumX Metrics
相关文献

 作者相关
 关键词相关
 参考文献相关

版权所有 ©2008 中国科学院文献情报中心 制作维护:中国科学院文献情报中心
地址:北京中关村北四环西路33号 邮政编码:100190 联系电话:(010)82627496 E-mail:cscd@mail.las.ac.cn 京ICP备05002861号-4 | 京公网安备11010802043238号